INT 131 - CAS 315224-26-1
Catalog number:
315224-26-1
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C21H12Cl4N2O3S
Molecular Weight:
511.93
COA:
Inquire
Targets:
PPAR
Description:
INT 131 is a hypoglycemic agent, displays robust glucose-lowering activity in rodent models of diabetes while exhibiting a reduced side-effects profile compared to marketed TZDs.
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Purity:
≥98%
Appearance:
Solid powder
Synonyms:
AMG 131; 2,4-Dichloro-N-(3,5-dichloro-4-quinolin-3-yloxyphenyl)benzenesulfonamide;
Solubility:
Soluble in DMSO
Storage:
Store at -20 °C
MSDS:
Inquire
Application:
Selective PPARgamma modulator, enhancing insulin sensitivity.
Quality Standard:
Enterprise standard
Shelf Life:
As supplied, 2 years from the QC date provided on the Certificate of Analysis, when stored properly.
Quantity:
Milligrams-Grams
InChIKey:
NMRWDFUZLLQSBN-UHFFFAOYSA-N
InChI:
1S/C21H12Cl4N2O3S/c22-13-5-6-20(16(23)8-13)31(28,29)27-14-9-17(24)21(18(25)10-14)30-15-7-12-3-1-2-4-19(12)26-11-15/h1-11,27H
Canonical SMILES:
C1=CC=C2C(=C1)C=C(C=N2)OC3=C(C=C(C=C3Cl)NS(=O)(=O)C4=C(C=C(C=C4)Cl)Cl)Cl
Current Developer:
InteKrin Therapeutics
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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