|Description||Indacaterol is an ultra-long-acting β-adrenoceptor agonist with pKi of 7.36.|
Vilanterol (GW642444; GW 642444X) is a novel, inhaled, long-acting β(2) agonist with inherent 24-h activity under development as a once-daily combination therap...
Timolol Maleate is a non-selective, beta-adrenergic receptor antagonist for β1/β2 with Ki of 1.97 nM/2.0 nM.
Betaxolol is a β1 adrenergic receptor blocker with IC50 of 6 μM.
Alfuzosin is a pharmaceutical drug of the alpha-1 blocker class. It works by relaxing the muscles in the prostate and bladder neck. It is used to treat benign p...
Etiguanfacine is a α2-Adreno Receptor agonist using for the treatment of ADHD (Attention deficit hyperactivity disorder).
ABT-866 is a novel alpha-adrenoceptor agent that demonstrates intrinsic activity at the α1A-adrenoceptor subtype present in the rabbit urethra (pD2=6.22, with 8...
(RS)-Butyryltimolol is the racemate of Butyryltimolol which is the butyryl ester of Timolol. Timolol, in the non-selective β blocker family of medication, has b...
The hydrochloride of Nifenalol. Nifenalol is a beta-adrenoceptor antagonist used for the treatment of cardiovascular and cerebrovascular diseases such as hypert...
Landiolol is an ultra-short-acting Beta 1 adrenergic receptor antagonist using for managing supraventricular tachyarrhythmias in sepsis. It is also used as an a...
Fenmetozole, also known as DH-524, is an antagonist of α2-adrenergic receptor and also antagonizes the actions of ethanol.
Fiduxosin is a potent antagonist of α1-adrenoceptor, with Ki= 0.160 nM, 24.9 nM, and 0.920 nM for α1a-, α1b-, and α1d-adrenoceptors, respectively. Fiduxosin was...
Salbutamol Sulfate is a Non-selective 2-adrenergic receptor agonist (IC50=8.93 µM)
Vilanterol, also known as GW-642444, is a long-acting beta-2 agonist drug, which in May 2013 was approved in combination with fluticasone furoate for sale as Br...
An α1 adrenergic receptor antagonist
Indacaterol is an ultra-long-acting β-adrenoceptor agonist with pKi of 7.36.
Metoprolol succinate is a selective β-adrenoceptor antagonist. It is used in treatment of several diseases of the cardiovascular system. It is a drug used in th...
P2647, also known as Benzquinamide, is a discontinued antiemetic compound with antihistaminic, mild anticholinergic, and sedative properties. P2647 binds to the...
Guanabenz Acetate is an selective agonist of α2a-adrenergic receptor, α2b-adrenergic receptor and α2c-adrenergic receptor with pEC50 of 8.25, 7.01 and ~5, respe...
Ritodrine HCl is a hydrochloride salt of ritodrine which is a β-2 adrenergic receptor agonist.Ritodrine (discontinued preparation: Yutopar) is a tocolytic drug,...
CP-114271, a thiazole derivative, has been found to be a β3 adrenergic receptor agonist that was once studied in obesity therapy.