INCB 3284 dimesylate - CAS 887401-93-6
Catalog number:
887401-93-6
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C26H31F3N4O4.2CH4O3S
Molecular Weight:
712.76
COA:
Inquire
Targets:
CCR
Description:
Potent, selective and orally bioavailable CCR2 antagonist with IC50 of 3.7 nM.
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Brife Description:
Potent, selective and orally bioavailable CCR2 antagonist with IC50 of 3.7 nM.
Appearance:
White to Off-White Solid
Synonyms:
N-[2-[[(3R)-1-[trans-4-hydroxy-4-(6-methoxy-3-pyridinyl)cyclohexyl]-3-pyrrolidinyl]amino]-2-oxoethyl]-3-(trifluoromethyl)-benzamide, dimethanesulfonate
Solubility:
DMSO: 42mg/mL;
Storage:
Store at -20°C
MSDS:
Inquire
Quality Standard:
In-house
Quantity:
Grams-Kilos
InChIKey:
PNPNUHKICDECDH-FBLZNNLISA-N
InChI:
1S/C26H31F3N4O4.2CH4O3S/c1-37-23-6-5-19(14-30-23)25(36)10-7-21(8-11-25)33-12-9-20(16-33)32-22(34)15-31-24(35)17-3-2-4-18(13-17)26(27,28)29;2*1-5(2,3)4/h2-6,13-14,20-21,36H,7-12,15-16H2,1H3,(H,31,35)(H,32,34);2*1H3,(H,2,3,4)/t20-,21-,25-;;/m1../
Canonical SMILES:
O[C@]1(C2=CN=C(OC)C=C2)CC[C@@H](N3C[C@H](NC(CNC(C4=CC(C(F)(F)F)=CC=C4)=O)=O)CC3)CC1.CS(=O)(O)=O.CS(=O)(O)=O
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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Chemical Structure

CAS 887401-93-6 INCB 3284 dimesylate

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