Impentamine dihydrobromide - CAS 149629-70-9
Category: Inhibitor
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Molecular Formula:
C8H17N3Br2
Molecular Weight:
315.05
COA:
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Targets:
Histamine Receptor
Description:
Impentamine dihydrobromide is the dihydrobromide salt of impentamine, which is a highly selective and the most potent histamine H3 antagonist with pA2 value of 8.4. It also acts as a partial agonist in SK-N-MC cells expressing human H3 receptors. It shows > 30000-fold selectivity over histamine H1 and H2 receptors.
Synonyms:
VUF 4702; VUF-4702; VUF4702; 4-(5-Aminopentyl)imidazole dihydrobromide
MSDS:
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InChIKey:
QSDXAAWBBPWGEL-UHFFFAOYSA-N
InChI:
InChI=1S/C8H15N3.2BrH/c9-5-3-1-2-4-8-6-10-7-11-8;;/h6-7H,1-5,9H2,(H,10,11);2*1H
Canonical SMILES:
C1=C(NC=N1)CCCCCN.Br.Br
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CAS 149629-70-9 Impentamine dihydrobromide

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