|Description||Impentamine dihydrobromide is the dihydrobromide salt of impentamine, which is a highly selective and the most potent histamine H3 antagonist with pA2 value of 8.4. It also acts as a partial agonist in SK-N-MC cells expressing human H3 receptors. It shows > 30000-fold selectivity over histamine H1 and H2 receptors.|
|Synonyms||VUF 4702; VUF-4702; VUF4702; 4-(5-Aminopentyl)imidazole dihydrobromide|
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