HG-9-91-01 - CAS 1456858-58-4
Catalog number:
1456858-58-4
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C32H37N7O3
Molecular Weight:
567.68
COA:
Inquire
Targets:
Ephrin Receptor | Salt-inducible Kinases (SIKs) | Src
Description:
HG-9-91-01,a small molecule inhibitor that targets specificly salt-inducible kinase (SIKs) IC50: SIK1=0.92 nM; SIK2=6.6 nM; SIK3=9.6 nM
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Appearance:
Solid powder
Synonyms:
1-(2,4-dimethoxyphenyl)-3-(2,6-dimethylphenyl)-1-[6-[4-(4-methylpiperazin-1-yl)anilino]pyrimidin-4-yl]urea HG-9-91-01 HY-15776 GTPL8049 SCHEMBL15271960 BDBM192712 CS-1749 HG-9-91-01 (1) 1-(2,4-dimethoxyphenyl)-3-(2,6-dimethylphenyl)-1-[6-[4-(4-methylpiper
Solubility:
Soluble to > 10 mM in DMSO
Storage:
Store in a cool and dry place and at 0 - 4℃ for short term (days to weeks) or -72℃ for long term (months to years).
MSDS:
Inquire
Shelf Life:
2 years
Quantity:
Grams-Kilos
Boiling Point:
790.8±60.0 °C | Condition: Press: 760 Torr
Density:
1.257±0.06 g/cm3
InChIKey:
UYUHRKLITDJEHB-UHFFFAOYSA-N
InChI:
1S/C32H37N7O3/c1-22-7-6-8-23(2)31(22)36-32(40)39(27-14-13-26(41-4)19-28(27)42-5)30-20-29(33-21-34-30)35-24-9-11-25(12-10-24)38-17-15-37(3)16-18-38/h6-14,19-21H,15-18H2,1-5H3,(H,36,40)(H,33,34,35)
Canonical SMILES:
CC1=C(C(=CC=C1)C)NC(=O)N(C2=C(C=C(C=C2)OC)OC)C3=NC=NC(=C3)NC4=CC=C(C=C4)N5CCN(CC5)C
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