GYKI-47261 - CAS 220445-20-5
Catalog number:
220445-20-5
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C18H15ClN4
Molecular Weight:
322.796
COA:
Inquire
Targets:
AMPAR
Description:
GYKI-47261 is a non-competitive AMPA receptor antagonist (IC50 = 2.5 μM) and a CYP2E1 inducer. GYKI-47261 shows broad spectrum anticonvulsive activity and neuroprotective effects in vivo.
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Purity:
>99 %
Appearance:
White to Off-White Solid
Synonyms:
4-(8-chloro-2-methyl-11H-imidazo[1,2-c][2,3]benzodiazepin-6-yl)aniline; GYKI 47261; GYKI-47261
MSDS:
Inquire
InChIKey:
FPXVCCSOTAQPIV-UHFFFAOYSA-N
InChI:
1S/C18H15ClN4/c1-11-10-23-17(21-11)8-13-2-5-14(19)9-16(13)18(22-23)12-3-6-15(20)7-4-12/h2-7,9-10H,8,20H2,1H3
Canonical SMILES:
CC1=CN2C(=N1)CC3=C(C=C(C=C3)Cl)C(=N2)C4=CC=C(C=C4)N
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CAS 220445-20-5 GYKI-47261

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