GYKI-46903 HCl - CAS 142999-59-5
Catalog number:
142999-59-5
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C17H21ClFNO2
Molecular Weight:
325.81
COA:
Inquire
Targets:
5-HT Receptor | mAChR
Description:
GYKI-46903 is a Muscarinic M3 receptor and Serotonin 3 receptor antagonist. In displacement studies, the pIC50 values of GYKI-46903 against [3H]granisetron binding to rat cerebral cortex membranes were 6.91. No development was reported for the treatment of Cognition disorders, Nausea and vomiting.
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Purity:
98%
Appearance:
Powder
Synonyms:
(4R,5R)-6-(4-fluorophenyl)-1-azabicyclo[3.3.1]non-6-en-4-yl propionate hydrochloride
Solubility:
Soluble in DMSO
Storage:
-20°C Freezer
MSDS:
Inquire
Application:
Cognition disorders; Nausea and vomiting
Quality Standard:
In-house standard
Shelf Life:
2 month in rt, long time
Quantity:
Milligrams-Grams
InChIKey:
UBIAWBSPCYNXMC-QNBGGDODSA-N
InChI:
1S/C17H20FNO2.ClH/c1-2-17(20)21-16-8-10-19-9-7-14(15(16)11-19)12-3-5-13(18)6-4-12;/h3-7,15-16H,2,8-11H2,1H3;1H/t15-,16-;/m1./s1
Canonical SMILES:
c1cc(ccc1F)C=1[C@@H]2[C@@H](CC[N@@](CC1)C2)OC(CC)=O.Cl
Current Developer:
Originator IVAX Drug Research Institute
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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