GYKI-14451 sulfate - CAS 83861-29-4
Catalog number:
83861-29-4
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C50-H76-N12-O10.H2-O4-S
Molecular Weight:
1103.30
COA:
Inquire
Targets:
Thrombin
Description:
GYKI-14451 is a synthetic tripeptide inhibitor of thrombin.It has anti-atherosclerotic activity.
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Purity:
98%
Appearance:
Powder
Synonyms:
tert-butyl ((R)-1-((S)-2-(((S)-5-guanidino-1-oxopentan-2-yl)carbamoyl)pyrrolidin-1-yl)-1-oxo-3-phenylpropan-2-yl)carbamate hemisulfate; LY 178207; Boc-D-Phe-Pro-Arg-H;69201-89-4 (free base)
Solubility:
Soluble in DMSO
Storage:
-20℃ Freezer
MSDS:
Inquire
Application:
Thrombosis
Quality Standard:
In-house standard
Shelf Life:
2 month in rt, long time
Quantity:
Milligrams-Grams
InChIKey:
KMQNMDPAZPATRK-DCBJEQAZSA-N
InChI:
1S/2C25H38N6O5.H2O4S/c2*1-25(2,3)36-24(35)29-19(15-17-9-5-4-6-10-17)21(33)30-22(34)20-12-8-14-31(20)18(16-32)11-7-13-28-23(26)27;1-5(2,3)4/h2*4-6,9-10,16,18-20H,7-8,11-15H2,1-3H3,(H,29,35)(H4,26,27,28)(H,30,33,34);(H2,1,2,3,4)/t2*18-,19+,20-;/m00./s1
Canonical SMILES:
CC(C)(C)OC(=O)N[C@H](Cc1ccccc1)C(=O)NC(=O)[C@@H]2CCCN2[C@@H](CCCNC(=N)N)C=O.CC(C)(C)OC(=O)N[C@H](Cc1ccccc1)C(=O)NC(=O)[C@@H]2CCCN2[C@@H](CCCNC(=N)N)C=O.OS(=O)(=O)O
Current Developer:
Originator IVAX Drug Research Institute
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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