GYKI 14166 - CAS 83997-16-4
Catalog number: 83997-16-4
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C20-H30-N6-O3.H2-O4-S
Molecular Weight:
500.57
COA:
Inquire
Targets:
Thrombin
Description:
Efegatran is a thrombin inhibitor under the development of Eli Lilly. It can be used for the treatment of thromboembolic disorders. No development reported was reported for the treatment of Thrombosis.
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Purity:
98%
Appearance:
Powder
Synonyms:
Efegatran;RGH2958; LY 294468; (S)-1-(D-phenylalanyl)-N-((S)-5-guanidino-1-oxopentan-2-yl)pyrrolidine-2-carboxamide sulfate
Solubility:
Soluble in DMSO
Storage:
-20℃ Freezer
MSDS:
Inquire
Application:
Thrombosis
Quality Standard:
In-house standard
Shelf Life:
2 month in rt, long time
Quantity:
Milligrams-Grams
InChIKey:
RMYMBMLRPYLYDX-VNMUXGFYSA-N
InChI:
1S/C20H30N6O3.H2O4S/c21-16(12-14-6-2-1-3-7-14)18(28)25-19(29)17-9-5-11-26(17)15(13-27)8-4-10-24-20(22)23;1-5(2,3)4/h1-3,6-7,13,15-17H,4-5,8-12,21H2,(H4,22,23,24)(H,25,28,29);(H2,1,2,3,4)/t15-,16+,17-;/m0./s1
Canonical SMILES:
c1ccc(cc1)C[C@H](C(=O)NC(=O)[C@@H]2CCCN2[C@@H](CCCNC(=N)N)C=O)N.OS(=O)(=O)O
Current Developer:
Eli Lilly
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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CAS 83997-16-4 GYKI 14166

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