|Description||GYKI-13324 is bifunctional nitrosoureido derivative and alkylating agent. It can produce long-term or total regression of adenomatous, but only marginal growth delay of mucinous tumors. GYKI-13324, seems to be a candidate in the clinical management of colorectal tumors.|
|Solubility||Soluble in DMSO|
|Quality Standard||In-house standard|
|Shelf Life||2 month in rt, long time|
Celgosivir, an effective α-glucosidase I inhibitor, has been found to be related to viral maturation and is still under Phase I/II trial against Dengue. IC50: 1...
Butylparaben is used as an antimicrobial preservative in cosmetics. It is also used in medication suspensions and used as a flavoring additive in food.
Warfarin is an anticoagulant applicated in the prevention of thrombosis and thromboembolism, the formation of blood clots in the blood vessels and their migrati...
Propylthiouracil is a thyroperoxidase and 5'-deiodinase inhibitor. It is a thiouracil-derived drug used to treat hyperthyroidism (including Graves' disease) by ...
Binfloxacin, a bio-active chemical compound, has antibiotic effect.
Rabeximod is an immunomodulator agent. It can suppress arthritis by preventing activation of inflammatory cells, most likely macrophages, in a time dependent fa...
Metaldehyde, the tetramer form of aldehyde, could be used in the production of other substances and also a pesticide against sorts of gastropods.
TOFA, also called as RMI14514 or MDL14514, is a cell-permeable, potent, reversible, and competitive allosteric inhibitor of acetyl-CoA carboxylase-α (ACCA). TOF...
RO5263397 is a selective trace amine-associated receptor 1(TAAR1) agonist. TAAR1 is a drug discovery target for cocaine addiction. RO5263397 is efficacious in r...
Neuromedin S (rat)
Neuromedin S, a novel neuropeptide of 36 amino acids isolated from rat brain as an endogenous ligand for the orphan G protein-coupled receptors FM-3/GPR66 and F...
Nedocromil is an inhaled anti-inflammatory agent for the preventive management of asthma.
NVP-231 is a potent, specific, and reversible CerK inhibitor that competitively inhibits binding of ceramide to CerK. NVP-231 is active in the low nanomolar ran...
G-36 is an antagonist of G protein-coupled estrogen receptor (GPER). It selectively inhibits estrogen-mediated activation of PI3-K by GPER and estrogen-mediated...
Nicotinic acid N-oxide
Nicotinic acid N-oxide is used to treat hyperlipoidemia.
Gadobutrol is a nonionic, paramagnetic contrast agent developed for tissue contrast enhancement in magnetic resonance imaging (MRI). It has a macrocyclic framew...
Bulleyaconitine A, an active indegrent from aconitum bulleyanum Diel, has been found to be effective in the treatment of chronic pain and rheumatoid arthritis.
CB-839 an is orally bioavailable inhibitor of glutaminase, with potential antineoplastic activity. Upon oral administration, CB-839 selectively and irreversibly...
Gastrin-Releasing Peptide, human
Gastrin-Releasing Peptide, human (GRP), one of the bombesin-like peptide family, is an agonist for the gastrin-releasing peptide receptor (GRPR) and it plays on...
Aloe-emodin is an interferon-inducing agent with IC50 of about 1 μg/mL for JEV and of about 0.33 μg/mL for EV71.
(±)-Epibatidine dihydrochloride is a highly potent nicotinic agonist used as a non-narcotic analgesic.