GW9508 - CAS 885101-89-3
Catalog number: B0084-272136
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C22H21NO3
Molecular Weight:
347.414
COA:
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Targets:
GPR40
Description:
GW9508 is a potent and selective agonist for FFA1 (GPR40) with pEC50 of 7.32, 100-fold selective against GPR120, and stimulates insulin secretion in a glucose-sensitive manner. GW9508 is commonly used in the treatment of type 2 diabetes.
Ordering Information
Catalog Number Size Price Stock Quantity
B0084-272136 100 mg $399 In stock
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Brife Description:
FFA1 (GPR40) agonist
Purity:
> 98%
Appearance:
Off-White to Pale Beige Solid
Synonyms:
GW-9508; GW 9508; 3-(4-((3-Phenoxybenzyl)amino)phenyl)propanoic acid
MSDS:
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Melting Point:
90-92°C
InChIKey:
DGENZVKCTGIDRZ-UHFFFAOYSA-N
InChI:
InChI=1S/C22H21NO3/c24-22(25)14-11-17-9-12-19(13-10-17)23-16-18-5-4-8-21(15-18)26-20-6-2-1-3-7-20/h1-10,12-13,15,23H,11,14,16H2,(H,24,25)
Canonical SMILES:
C1=CC=C(C=C1)OC2=CC=CC(=C2)CNC3=CC=C(C=C3)CCC(=O)O
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CAS 885101-89-3 GW9508

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