GV-58 - CAS 1402821-41-3
Catalog number: 1402821-41-3
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C18H26N6OS
Molecular Weight:
374.50
COA:
Inquire
Targets:
Calcium Channel
Description:
GV-58, a pupin derivative, has been found to be a P/Q-type Ca²⁺-channel agonist that could be used to against neuromuscular weakness. IC50: 7.21/8.81 uM (N-type/P-Q-type Ca2+ channel).
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Purity:
98%
Appearance:
Powder
Synonyms:
GV-58; CHEMBL2206242; SCHEMBL17628602; BDBM50400564; CS-3617
Solubility:
10 mM in DMSO
Storage:
-20ºC Freeze
MSDS:
Inquire
Application:
GV-58 has been found to be a P/Q-type Ca²⁺-channel agonist that could be used to against neuromuscular weakness.
Shelf Life:
As supplied, 2 years from the QC date provided on the Certificate of Analysis, when stored properly
Quantity:
Millgrams-Grams
InChIKey:
DPTXJOUVBMUSGY-CYBMUJFWSA-N
InChI:
InChI=1S/C18H26N6OS/c1-4-8-24-11-20-15-16(19-9-14-7-6-12(3)26-14)22-18(23-17(15)24)21-13(5-2)10-25/h6-7,11,13,25H,4-5,8-10H2,1-3H3,(H2,19,21,22,23)/t13-/m1/s1
Canonical SMILES:
CCCN1C=NC2=C1N=C(N=C2NCC3=CC=C(S3)C)NC(CC)CO
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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