Gue 1654 - CAS 397290-30-1
Category: Inhibitor
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Molecular Formula:
C23H17N3OS3
Molecular Weight:
447.6
COA:
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Targets:
Others
Description:
Gue 1654 is an oxoeicosanoid receptor 1 (OXE-R) modulator selectively inhibiting Gβγ but not Gαi signaling upon activation of the Gαi-βγ heterotrimer by OXE-R. Gue 1654 was shown to inhibit Gβγ-mediated opening of GIRK1/2 channels in HEK293 cells.
Brife Description:
OXE-R modulator
Purity:
≥97% by HPLC
Synonyms:
Gue1654; Gue 1654; Gue-1654. N-[7-(Methylthio)benzo[1,2-d:4,3-d']bisthiazol-2-yl]-α-phenylbenzeneacetamide
MSDS:
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InChIKey:
UFOBDFMYJABXGK-UHFFFAOYSA-N
InChI:
InChI=1S/C23H17N3OS3/c1-28-23-25-17-13-12-16-19(20(17)30-23)29-22(24-16)26-21(27)18(14-8-4-2-5-9-14)15-10-6-3-7-11-15/h2-13,18H,1H3,(H,24,26,27)
Canonical SMILES:
CSC1=NC2=C(S1)C3=C(C=C2)N=C(S3)NC(=O)C(C4=CC=CC=C4)C5=CC=CC=C5
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Chemical Structure

CAS 397290-30-1 Gue 1654

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