|Description||Guanoxabenz, a metabolite of guanaben, is an α2 adrenergic receptor agonist.|
|Synonyms||2-[(E)-(2,6-dichlorophenyl)methylideneamino]-1-hydroxyguanidine; 1-(2,6-dichlorobenzylideneamino)-3-hydroxyguanidine; guanoxabenz; guanoxabenz hydrochloride; guanoxabenz monohydrochloride|
|Storage||Store in a cool and dry place (or refer to the Certificate of Analysis).|
|Boiling Point||383.1±52.0 ℃ at 760 Torr|
Terbutaline, also called as Bronclyn, as a fast-acting bronchodilator it is a β2 adrenergic receptor agonist used to treat asthma and premature labor.
Pronethalol is a non-selective beta-adrenergic blocking agentused in treatment due to carcinogenic properties.
Terazosin, works by blocking the action of adrenaline on smooth muscle of the bladder and the blood vessel walls, is a selective alpha1-antagonist used for trea...
Aptazapine is a tetracyclic antidepressant. It was assayed in clinical trials for the treatment of depression in the 1980s but was never marketed. Aptazapine is...
AR-08 is an agonist of α2-adrenergic receptor undergone in phase II clinical trials by Arbor Pharmaceuticals for the treatment of attention deficit and hyperac...
Guanabenz Acetate is an selective agonist of α2a-adrenergic receptor, α2b-adrenergic receptor and α2c-adrenergic receptor with pEC50 of 8.25, 7.01 and ~5, respe...
Octopamine hydrochloride is an α-adrenoceptor agonist.
Carmoterol, a quinolin derivative, has been found to a β2-adrenoceptor agonist that could be an effective bronchodilating agent.
CL-316243 is a highly selective β3-adrenoceptor agonist with EC50 value of 3 nM; > 10000-fold selective over β1 and β2 receptors. CL-316243 can restore the expr...
QF0301B is an α1 adrenergic receptor antagonist and shows noncompetitive low action in 5-HT3, muscarinic and nicotinic receptors, or as Ca2+ antagonist.
Yohimbine, an indolalkylamine alkaloid, blocks presynaptic alpha-2 adrenergic receptors. IC50= 0.6 μM Ki: 1.05 nM, alphaα2Areceptor
Rezatomidine is a selective α2-adrenoreceptor antagonist under the development of Allergan. No recent development was reported for the treatment of Diabetic neu...
Falintolol, (Z)- is a novel β-adrenergic antagonist.
Levonordefrin is a adrenergic receptor agonist and can be used as a topical nasal decongestant and vasoconstrictor in dentistry in the United States. Levonordef...
MK-0634, also called as L-796568, is an β3 adrenergic receptor agonist that was progressed into clinical studies for the treatment of obesity in the early 2000s...
Prazosin, a selective and orally active antagonist of adrenergic alpha-1, is a synthetic piperazine derivative to treat high blood pressure and anxiety, PTSD, a...
SNAP-8719, structurally very similar to BMY-7378, is a selective, orally active α1D-AR antagonist with lower binding affinity for the 5-HT1A receptor.
Medetomidine is a selective α2-adrenoceptor agonist, with Ki of 1.08 nM, exhibts 1620-fold selectivity over α1-adrenoceptor.
CP-114271, a thiazole derivative, has been found to be a β3 adrenergic receptor agonist that was once studied in obesity therapy.
Nifenalol, also known as INPEA, is a novel antagonist of β-adrenoceptors.