|Description||GSK894490A is a non-peptide ghrelin receptor agonist. It crosses the blood/brain barrier and elicit pro-cognitive effects in recognition and spatial learning and memory tests. It may be used as a potential drug target for therapeutic approaches to treat diseases affecting cognition.|
|Synonyms||Benzenesulfonamide, N-(5-((3R,5S)-3,5-dimethyl-1-piperazinyl)-2-methoxyphenyl)-4-(5-methyl-2-furanyl)-, hydrochloride (1:1), rel-;N-[5-[(3R,5S)-3,5-dimethylpiperazin-1-yl]-2-methoxyphenyl]-4-(5-methylfuran-2-yl)benzenesulfonamide hydrochloride;GSK-894490A|
|Solubility||10 mM in DMSO|
|Application||GSK894490A may be used as a potential drug target for therapeutic approaches to treat diseases affecting cognition.|
|Quality Standard||In-house standard|
|Shelf Life||2 month in rt, long time|
Noradrenaline bitartrate monohydrate
Noradrenaline bitartrate monohydrate is a direct alpha-adrenergic receptors stimulator.Noradrenaline modulates the gain of evoked activity, especially in sensor...
Bendroflumethiazide is a thiazide diuretic as a Na++Cl- symport inhibitor. Bendroflumethiazide can be used in the treatment of mild heart failure although loop ...
GYY-4137 Morpholine salt
GYY-4137 Morpholine salt is a novel water-soluble and slow releasing Hydrogen sulfide(H2S) donor. It protects against myocardial ischemia and reperfusion injury...
Glafenine is a non-steroidal analgesic agent, shows significant antiinflammatory activity.
Aminocaproic acid is a derivative and analogue of the amino acid lysine, which makes it an effective inhibitor for enzymes that bind that particular residue. Su...
EPZ020411, with potent anticancer activity, is an orally bioactive, selective inhibitor of PRMT6/8/1 with over 100-fold selective for other histone methyltransf...
Schisandrol B is one of its major active constituents of traditional hepato-protective Chinese medicine, Schisandra sphenanthera.
Metyrapol, a dipyridine derivative, has been found to be a 11-deoxycorticosterone hydroxylation inhibitor and could always used as a medical diagnostic reagent ...
Trimetazidine dihydrochloride, a piperazine derivative, could reduce fatty acid β-oxidation and used as a coronary vasodilator.
Gadoteridol, a MRI contrast agent, is commonly used in central nervous system imaging.
Tetrahydrofolic acid is a folic acid derivative. It is a cofactor in many bio-reactions, especially in the metabolism of amino acids and nucleic acids.
Hemoglobin Modulators-1, a substituted benzaldehyde compound that can modulate sickle hemoglobin (HbS) for treatment of disorders.
DO3A tert-Butyl ester
DOTA tert-Butyl ester is a benxyl derivative of the cyclic tosamide; can be nitrated directly; is more convenient to incorporate the nitro group after deprotect...
Microorganisms commonly accumulate at interfaces as part of biofilms held together by a matrix of hydrated extracellular polymeric substances. cis-2-Decenoic ac...
CC-17368, a hydroxyisoindole derivative, is a metabolites of pomalidomide and has potential activity in anticancer study like multiple myeloma.
Osilodrostat, also called as LCI699, is a modulator of 11-β-hydroxylase (IC50= 2.5 nM), useful for treating a disorder ameliorated 11-β-hydroxylase inhibition, ...
Chlorpropamide is a drug in the sulfonylurea class used to treat type 2 diabetes mellitus. It is a long-acting 1st generation sulfonylurea.
Bufalin is a major digoxin-like immunoreactive component of the Chinese medicine Chan Su and has been shown to exert a potential for anticancer activity against...
Tocainide, a lidocaine analog, is a class Ib antiarrhythmic agent.
CP-71362 is a pentapeptide renin inhibitor. It is selective for the canine enzyme.