GSK7227 - CAS 1067214-81-6
Catalog number: 1067214-81-6
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C25H22N2O6S
Molecular Weight:
478.52
COA:
Inquire
Targets:
PPAR
Description:
GSK7227 is a novel class of PPARdelta partial agonists. It shows potent partial agonism of the PPARdelta target genes CPT1a and PDK4 in skeletal muscle cells.
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Purity:
>98%
Appearance:
Solid powder
Synonyms:
2-[[3-(5-Methoxy-4-methylindol-1-yl)sulfonylbenzoyl]amino]-5-methylbenzoic acid;GSK-7227;Benzoic acid, 2-((3-((5-methoxy-4-methyl-1H-indol-1-yl)sulfonyl)benzoyl)amino)-5-methyl-
Solubility:
10 mM in DMSO
Storage:
-20°C Freezer
MSDS:
Inquire
Quality Standard:
In-house standard
Shelf Life:
2 month in rt, long time
Quantity:
Milligrams-Grams
Density:
1.35±0.1 g/cm3 | Condition: Temp: 20 °C Press: 760 Torr
InChIKey:
LYXBTAXWNCLYLA-UHFFFAOYSA-N
InChI:
InChI=1S/C25H22N2O6S/c1-15-7-8-21(20(13-15)25(29)30)26-24(28)17-5-4-6-18(14-17)34(31,32)27-12-11-19-16(2)23(33-3)10-9-22(19)27/h4-14H,1-3H3,(H,26,28)(H,29,30)
Canonical SMILES:
CC1=CC(=C(C=C1)NC(=O)C2=CC(=CC=C2)S(=O)(=O)N3C=CC4=C3C=CC(=C4C)OC)C(=O)O
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