GSK4112 - CAS 1216744-19-2
Catalog number: 1216744-19-2
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C18H21ClN2O4S
Molecular Weight:
396.89
COA:
Inquire
Targets:
Others
Description:
GSK 4112, a kind of synthetic agonist of REV-ERBα, could suppress the expression of sorts of genes involved in gluconeogenesis. IC50: 0.4 μM (EC50).
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Purity:
95%
Appearance:
Powder
Synonyms:
GSK4112;SR6452;CHEMBL1961795;1216744-19-2;MLS006010708;GTPL2903
Solubility:
10 mM in DMSO
Storage:
-20ºC Freeze
MSDS:
Inquire
Application:
GSK 4112 is a kind of synthetic agonist of REV-ERBα and could suppress the expression of sorts of genes involved in gluconeogenesis.
Shelf Life:
As supplied, 2 years from the QC date provided on the Certificate of Analysis, when stored properly
Quantity:
Milligrams-Grams
InChIKey:
WYSLOKHVFKLWOU-UHFFFAOYSA-N
InChI:
InChI=1S/C18H21ClN2O4S/c1-18(2,3)25-17(22)12-20(10-13-4-6-14(19)7-5-13)11-15-8-9-16(26-15)21(23)24/h4-9H,10-12H2,1-3H3
Canonical SMILES:
CC(C)(C)OC(=O)CN(CC1=CC=C(C=C1)Cl)CC2=CC=C(S2)[N+](=O)[O-]
Current Developer:
GSK
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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Chemical Structure

CAS 1216744-19-2 GSK4112

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