GSK2330672 - CAS 1345982-69-5
Catalog number:
1345982-69-5
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C28H38N2O7S
Molecular Weight:
546.68
COA:
Inquire
Targets:
Others
Description:
GSK-2330672, an ASBT inhibitor, has been developed for the treatment of type 2 diabetes and is currently under Phase II trail against primary biliary cirrhosis and type 2 diabetes. IC50: 42 ± 3 nM.
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Purity:
98%
Appearance:
Powder
Synonyms:
CHEMBL2387408; UNII-386012Z45S; GSK2330672; GSK-2330672; SCHEMBL2586025; CZGVOBIGEBDYTP-VSGBNLITSA-N
Solubility:
DMSO: ≥ 21.5 mg/mL
Storage:
-20ºC Freeze
MSDS:
Inquire
Application:
GSK-2330672 is an ASBT inhibitor that has been developed for the treatment of type 2 diabetes and is currently under Phase II trail against primary biliary cirrhosis and type 2 diabetes.
Shelf Life:
As supplied, 2 years from the QC date provided on the Certificate of Analysis, when stored properly
Quantity:
Milligrams-Grams
InChIKey:
CZGVOBIGEBDYTP-VSGBNLITSA-N
InChI:
InChI=1S/C28H38N2O7S/c1-4-6-12-28(5-2)18-38(35,36)24-13-20(17-29-21(14-25(31)32)15-26(33)34)23(37-3)16-22(24)27(30-28)19-10-8-7-9-11-19/h7-11,13,16,21,27,29-30H,4-6,12,14-15,17-18H2,1-3H3,(H,31,32)(H,33,34)/t27-,28-/m1/s1
Canonical SMILES:
CCCCC1(CS(=O)(=O)C2=CC(=C(C=C2C(N1)C3=CC=CC=C3)OC)CNC(CC(=O)O)CC(=O)O)CC
Current Developer:
GSK
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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