GSK2269557 - CAS 1254036-71-9
Catalog number:
1254036-71-9
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C26H28N6O
Molecular Weight:
440.54
COA:
Inquire
Targets:
PI3K
Description:
GSK2269557, an effective PI3K inhibitor, could be used as against inflammatory and some autoimmune diseases. It has just completes a phase II trial against Asthma.
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Purity:
95%
Appearance:
Powder
Synonyms:
CHEMBL2216859; GSK2269557 (free base); GSK-2269557; 2-(6-(1H-indol-4-yl)-1H-indazol-4-yl)-5-((4-isopropylpiperazin-1-yl)methyl)oxazole; 6-(1H-indol-4-yl)-4-(5-{[4-(1-methylethyl)-1-piperazinyl]methyl}-1,3-oxazol-2-yl)-1H-indazole
Solubility:
DMSO
Storage:
-20ºC Freeze
MSDS:
Inquire
Application:
GSK2269557 is an effective PI3K inhibitor that could be used as against inflammatory and some autoimmune diseases.
Shelf Life:
As supplied, 2 years from the QC date provided on the Certificate of Analysis, when stored properly
Quantity:
Milligrams-Grams
InChIKey:
MCIDWGZGWVSZMK-UHFFFAOYSA-N
InChI:
InChI=1S/C26H28N6O/c1-17(2)32-10-8-31(9-11-32)16-19-14-28-26(33-19)22-12-18(13-25-23(22)15-29-30-25)20-4-3-5-24-21(20)6-7-27-24/h3-7,12-15,17,27H,8-11,16H2,1-2H3,(H,29,30)
Canonical SMILES:
CC(C)N1CCN(CC1)CC2=CN=C(O2)C3=C4C=NNC4=CC(=C3)C5=C6C=CNC6=CC=C5
Current Developer:
GSK
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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