|Description||GSK'872 is aRIPK3inhibitor, which binds RIP3 kinase domain with high affinity (IC50=1.8 nM), and is approximately >1,000-fold selective over 300 kinases in a fluorescence polarization assay at a concentration of 1 μM. Besides, GSK'872 inhibits kinase activity (IC50=1.3 nM).|
|Brife Description||An inhibitor of receptor interacting protein kinase-3 (RIP3)|
|Solubility||DMSO: ≥ 150 mg/mL|
|Storage||Store in a cool and dry place (or refer to the Certificate of Analysis).|
|Boiling Point||625.7±55.0 ℃ at 760 Torr|
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