GSK-598809 - CAS 1310803-30-5
Catalog number: 1310803-30-5
Category: Inhibitor
Please be kindly noted products are not for therapeutic use. We do not sell to patients.
Molecular Formula:
C23H25F4N5OS
Molecular Weight:
495.54
COA:
Inquire
Targets:
Dopamine Receptor
Description:
GSK598809 is a selective Dopamine D3 receptor antagonist originated by GlaxoSmithKline. It may decrease the rewarding effects of contextual cues associated with drug intake preclinically and that may reduce drug craving in humans. No recent development for the treatment of Drug abuse. Eating disorders and Smoking withdrawal was reported.
Purity:
98%
Appearance:
Powder
Synonyms:
GSK-598809; GSK 598809; GSK598809; NII-Y5OZ63HC3V;5-(5-((3-((1S,5R)-1-(2-Fluoro-4-(trifluoromethyl)phenyl)-5-methyl-3-azabicyclo(3.1.0)hexan-3-yl)propyl)thio)-4-methyl-4H-1,2,4-triazol-3-yl)-4-methyloxazole
Solubility:
Soluble in DMSO
Storage:
-20°C Freezer
MSDS:
Inquire
Application:
Drug abuse; Eating disorders; Smoking withdrawal
Quality Standard:
In-house standard
Shelf Life:
2 month in rt, long time
Quantity:
Milligrams-Grams
InChIKey:
BAFWBNHYBAXTSE-FCHUYYIVSA-N
InChI:
1S/C23H25F4N5OS/c1-14-18(33-13-28-14)19-29-30-20(31(19)3)34-8-4-7-32-11-21(2)10-22(21,12-32)16-6-5-15(9-17(16)24)23(25,26)27/h5-6,9,13H,4,7-8,10-12H2,1-3H3/t21-,22+/m0/s1
Canonical SMILES:
Cc1c(ocn1)c2nnc(n2C)SCCCN3C[C@@]4(C[C@@]4(C3)c5ccc(cc5F)C(F)(F)F)C
Current Developer:
GlaxoSmithKline
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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