|Description||GSK 4716 is a selective agonist of estrogen-related receptors ERRβ and ERRγ displaying selectivity over ERRα and the classical estrogen receptors. Activation of GSK 4716 regulates mitochondrial activity in skeletal muscle during exercise.|
|Brife Description||ERRβ/γ agonist|
|Purity||≥99% by HPLC|
(R)-DPN has been found to be an estrogen receptor (ER) β agonist with higher affinity for estrogen receptor.
Ethisterone is a progestogen hormone being considered to treat prostate cancer.It was the first orally-active progestin.
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Raloxifene is an oral selective estrogen receptor modulator (SERM) that has estrogenic actions on bone and anti-estrogenic actions on the uterus and breast. It ...
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Tamoxifen Citrate is an antagonist of the estrogen receptor by competitive inhibition of estrogen binding, leading to a reduction in DNA synthesis and cellular ...
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Pipendoxifene hydrochloride is the hydrochloride salt of Pipendoxifene which
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Genistin is a derivative of Genistein, which is a PTK inhibitor. Genistin acts as a selective estrogen receptor modulator (SERM). It increases growth of breast ...