GSK-2881078 - CAS 1539314-06-1
Catalog number: 1539314-06-1
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C14H13F3N2O2S
Molecular Weight:
330.33
COA:
Inquire
Targets:
Androgen Receptor
Description:
GSK-2881078, an indole derivative, has been found to be an androgen receptor modulator that could probably be effective against Cachexia. It is still under Phase I trail.
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Purity:
98%
Appearance:
Powder
Synonyms:
GSK-2881078; SCHEMBL15421613; SKDVMPZQJMZEAC-SECBINFHSA-N; CS-5736; (R)-1-(1-(methylsulfonyl)propan-2-yl)-4-(trifluoromethyl)-1H-indole-5-carbonitrile
Solubility:
DMSO: ≥ 33 mg/mL
Storage:
Store in a cool and dry place and at 0 - 4 °C for short term (days to weeks) or -20 °C for long term (months to years).
MSDS:
Inquire
Quality Standard:
In-house standard
Quantity:
Milligram-Grams
InChIKey:
SKDVMPZQJMZEAC-SECBINFHSA-N
InChI:
InChI=1S/C14H13F3N2O2S/c1-9(8-22(2,20)21)19-6-5-11-12(19)4-3-10(7-18)13(11)14(15,16)17/h3-6,9H,8H2,1-2H3/t9-/m1/s1
Canonical SMILES:
CC(CS(=O)(=O)C)N1C=CC2=C1C=CC(=C2C(F)(F)F)C#N
Current Developer:
GSK
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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