GSK-239512 - CAS 720691-69-0
Catalog number:
720691-69-0
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C23H27N3O2
Molecular Weight:
377.48
COA:
Inquire
Targets:
Histamine Receptor
Description:
GSK-239512 is a histamine H3 receptor antagonist. In Jun 2015, Phase-II for Schizophrenia in USA was discontinued. Phase II clinical trilas for the treatment of Multiple sclerosis are on-going.
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Purity:
98%
Appearance:
Powder
Synonyms:
1-(6-((3-cyclobutyl-2,3,4,5-tetrahydro-1H-3-benzazepin-7-yl)oxy)-3-pyridinyl)-2-Pyrrolidinone
Solubility:
Soluble in DMSO
Storage:
-20℃ Freezer
MSDS:
Inquire
Application:
Multiple sclerosis
Quality Standard:
In-house standard
Shelf Life:
2 month in rt, long time
Quantity:
Milligrams-Grams
InChIKey:
YFRBKEVUUCQYOW-UHFFFAOYSA-N
InChI:
1S/C23H27N3O2/c27-23-5-2-12-26(23)20-7-9-22(24-16-20)28-21-8-6-17-10-13-25(19-3-1-4-19)14-11-18(17)15-21/h6-9,15-16,19H,1-5,10-14H2
Canonical SMILES:
O=C1CCCN1c2ccc(Oc3ccc4CCN(CCc4c3)C5CCC5)nc2
Current Developer:
Originator GlaxoSmithKline
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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