GSK-1440115 - CAS 1003878-16-7
Catalog number:
1003878-16-7
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C30H29Cl2N3O6
Molecular Weight:
598.47
COA:
Inquire
Targets:
Others
Description:
GSK-1440115 is an orally active urotensin II receptor antagonist. It is used for the treatment of asthma.
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Purity:
>98 %
Appearance:
Solid powder
Synonyms:
GSK1440115;4'-(1-(((6,7-Dichloro-3-oxo-2,3-dihydro-4H-1,4-benzoxazin-4-yl)acetyl)(methyl)amino)-2-(4-morpholinyl)ethyl)-4-diphenylcarboxylic acid;4-[4-[(1R)-1-[[2-(6,7-dichloro-3-oxo-1,4-benzoxazin-4-yl)acetyl]-methylamino]-2-morpholin-4-ylethyl]phenyl]benzoic acid
Solubility:
10 mM in DMSO
Storage:
-20°C Freezer
MSDS:
Inquire
Application:
GSK-1440115 is used for the treatment of asthma.
Quality Standard:
In-house standard
Shelf Life:
2 month in rt, long time
Quantity:
Milligrams-Grams
Melting Point:
858.9±65.0 °C | Condition: Press: 760 Torr
Density:
1.378±0.06 g/cm3 | Condition: Temp: 20 °C Press: 760 Torr
InChIKey:
YNBJTYUXPHTSFF-SANMLTNESA-N
InChI:
InChI=1S/C30H29Cl2N3O6/c1-33(28(36)17-35-25-14-23(31)24(32)15-27(25)41-18-29(35)37)26(16-34-10-12-40-13-11-34)21-6-2-19(3-7-21)20-4-8-22(9-5-20)30(38)39/h2-9,14-15,26H,10-13,16-18H2,1H3,(H,38,39)/t26-/m0/s1
Canonical SMILES:
CN(C(CN1CCOCC1)C2=CC=C(C=C2)C3=CC=C(C=C3)C(=O)O)C(=O)CN4C(=O)COC5=CC(=C(C=C54)Cl)Cl
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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