GSK-1070916A - CAS 942918-07-2
Catalog number:
942918-07-2
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
COA:
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Targets:
Aurora Kinase
Description:
GSK-1070916A is an ATP-competitive inhibitor of the serine/threonine kinases Aurora B and C with potential antineoplastic activity. Aurora B/C kinase inhibitor GSK1070916A binds to and inhibits the activity of Aurora kinases B and C, which may result in inhibition of cellular division and a decrease in the proliferation of tumor cells that overexpress the Aurora kinases B and C. Aurora kinases play essential roles in mitotic checkpoint control during mitosis, and are overexpressed by a wide variety of cancer cell types.
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Synonyms:
GSK-1070916A; GSK1070916A; GSK 1070916A.
MSDS:
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Current Developer:
GlaxoSmithKline, Inc.
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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CAS 942918-07-2 GSK-1070916A

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