GS 39783 - CAS 39069-52-8
Catalog number: 39069-52-8
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C15H23N5O2S
Molecular Weight:
337.44
COA:
Inquire
Targets:
GABA Receptor
Description:
GS 39783 is an allosteric positive modulator of GABAB receptors, decreases cocaine self-administration, blocks the rewarding properties of nicotine and produces anxiolytic-like activity without the side effects associated with baclofen or benzodiazepines.
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Purity:
≥98%
Appearance:
Pale orange solid
Synonyms:
N,N'-Dicyclopentyl-2-(methylthio)-5-nitro-4,6-pyrimidinediamine;4-N,6-N-dicyclopentyl-2-methylsulfanyl-5-nitropyrimidine-4,6-diamine;
Solubility:
Soluble in DMSO
Storage:
Store at -20 °C
MSDS:
Inquire
Application:
Positive allosteric modulator of GABAB receptor function.
Quality Standard:
Enterprise standard
Shelf Life:
As supplied, 2 years from the QC date provided on the Certificate of Analysis, when stored properly.
Quantity:
Milligrams-Grams
InChIKey:
GSGVDKOCBKBMGG-UHFFFAOYSA-N
InChI:
1S/C15H23N5O2S/c1-23-15-18-13(16-10-6-2-3-7-10)12(20(21)22)14(19-15)17-11-8-4-5-9-11/h10-11H,2-9H2,1H3,(H2,16,17,18,19)
Canonical SMILES:
CSC1=NC(=C(C(=N1)NC2CCCC2)[N+](=O)[O-])NC3CCCC3
Current Developer:
Gilead Sciences
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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