|Description||GS 39783 is an allosteric positive modulator of GABAB receptors, decreases cocaine self-administration, blocks the rewarding properties of nicotine and produces anxiolytic-like activity without the side effects associated with baclofen or benzodiazepines.|
|Appearance||Pale orange solid|
|Solubility||Soluble in DMSO|
|Storage||Store at -20 °C|
|Application||Positive allosteric modulator of GABAB receptor function.|
|Quality Standard||Enterprise standard|
|Shelf Life||As supplied, 2 years from the QC date provided on the Certificate of Analysis, when stored properly.|
|Current Developer||Gilead Sciences|
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