GR 79236 - CAS 124555-18-6
Catalog number:
124555-18-6
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C15H21N5O5
Molecular Weight:
351.36
COA:
Inquire
Targets:
Adenosine Receptor
Description:
GR 79236, an effective Adenosine A1 receptor agonist, could probably be used as an anti-inflammatory agent. IC50: 3.1 nM(Ki).
Publictions citing BOC Sciences Products
  • >> More
Purity:
95%
Appearance:
White solid
Synonyms:
N-[(1S, trans)-2-Hydroxycyclopentyl]adenosine
Solubility:
100 mM in H2O
Storage:
-20ºC Freeze
MSDS:
Inquire
Application:
GR 79236 is an effective Adenosine A1 receptor agonist that could probably be used as an anti-inflammatory agent.
Shelf Life:
As supplied, 2 years from the QC date provided on the Certificate of Analysis, when stored properly
Quantity:
Milligrams-Grams
Boiling Point:
728.3ºC at 760mmHg
Density:
1.89g/cm3
InChIKey:
GYWXTRVEUURNEW-QPIWWKSXSA-N
InChI:
InChI=1S/C15H21N5O5/c21-4-9-11(23)12(24)15(25-9)20-6-18-10-13(16-5-17-14(10)20)19-7-2-1-3-8(7)22/h5-9,11-12,15,21-24H,1-4H2,(H,16,17,19)/t7-,8-,9+,11?,12-,15+/m0/s1
Canonical SMILES:
C1CC(C(C1)O)NC2=NC=NC3=C2N=CN3C4C(C(C(O4)CO)O)O
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

Related Adenosine Receptor Products


CAS 1246018-36-9 ST4206

ST4206
(CAS: 1246018-36-9)

ST4206 is a potent adenosine A2A antagonist. ST4206 showed neuroprotective effects against rotenone induced alterations instriatal slice preparations,supporting...

CAS 152918-26-8 AB-MECA

AB-MECA
(CAS: 152918-26-8)

AB-MECA, a adenosine derivative, is a high affinity human A3 receptor in HEK 293 cells agonist.

CAS 53885-35-1 Ticlopidine Hydrochloride

Ticlopidine Hydrochloride
(CAS: 53885-35-1)

Ticlopidine HCl is an P2 receptor inhibitor against ADP-induced platelet aggregation with IC50 of ~2 μM.

CAS 1202402-40-1 CPI-444

CPI-444
(CAS: 1202402-40-1)

CPI-444 is a potent, orally available, selective antagonist of the adenosine A2A receptor that has been well tolerated in Ph 1/1b studies in non-oncology indica...

CAS 96392-15-3 PD-117519

PD-117519
(CAS: 96392-15-3)

PD-117519 is a N6-substituted adenosine receptor agonist. It shows oral antihypertensive activity in pharmacological animal models. It is used as a potential an...

Trabodenoson
(CAS: 871108-05-3)

Trabodenoson is a selective adenosine A1 receptor agonist. Trabodenoson can significantly reduce IOP in glaucoma and OHT patients. Phase III clinical trials for...

CGS 21680
(CAS: 120225-54-9)

CGS 21680, an A2 adenosine receptor selective agonist, has been found to be probably effective in inducing vasorelaxation and increasing in heart rate.

CAS 163838-04-8 UP202-56

UP202-56
(CAS: 163838-04-8)

UP202-56, an adenosine analogue, selectively acts via A1 receptors to significantly decrease noxiously-evoked spinal c-Fos protein expression.

CAS 544417-40-5 Capadenoson

Capadenoson
(CAS: 544417-40-5)

Capadenoson is a potent and selective adenosine A1 receptor agonist, which is a powerful protective mechanism in cerebral.

CAS 124431-80-7 CGS 21680 Hydrochloride

CGS 21680 Hydrochloride
(CAS: 124431-80-7)

CGS 21680 Hcl is an adenosine A2 receptor agonist with IC50 of 22 nM, exhibits 140-fold over A1 receptor.

CAS 479-18-5 Dyphylline

Dyphylline
(CAS: 479-18-5)

Dyphylline is a xanthine derivative with bronchodilator and vasodilator effects.It is used in the treatment of respiratory disorders like asthma, cardiac dyspne...

CAS 870070-55-6 Tozadenant

Tozadenant
(CAS: 870070-55-6)

An orally administered, potent and selective inhibitor of the adenosine 2a (A2a) receptor

CAS 36396-99-3 N6-Cyclohexyladenosine

N6-Cyclohexyladenosine
(CAS: 36396-99-3)

N6-Cyclohexyladenosine is a derivative of Adenosine, a selective A1 receptor agonist with EC50 = 8.2 nM.

CVT5440
(CAS: 531506-64-6)

CVT5440 is a selective, high affinity A(2B) adenosine receptor antagonist. It may has the potential treatment of asthma and has good selectivity.

CAS 131865-88-8 Sonedenoson

Sonedenoson
(CAS: 131865-88-8)

Sonedenoson is an adenosine A2 receptor agonist under the development of King Pharmaceuticals Research and Development. It can effectively promote rapid wound h...

CAS 28822-58-4 IBMX

IBMX
(CAS: 28822-58-4)

Non-specific inhibitor of cAMP and cGMP phosphodiesterases. The increase in cAMP level as a result of phosphodiesterase inhibition by IBMX activates PKA leading...

CAS 124555-18-6 GR 79236

GR 79236
(CAS: 124555-18-6)

GR 79236, an effective Adenosine A1 receptor agonist, could probably be used as an anti-inflammatory agent. IC50: 3.1 nM(Ki).

CAS 139180-30-6 ZM 241385

ZM 241385
(CAS: 139180-30-6)

Potent, highly selective A2A antagonist

CAS 58-55-9 Theophylline

Theophylline
(CAS: 58-55-9)

Theophylline is a methylated xanthine derivative; that functions as a nonselective PDE4 inhibitor and nonselective adenosine receptor antagonist.

CAS 20125-39-7 N6-(2-Phenylethyl)adenosine

N6-(2-Phenylethyl)adenosine
(CAS: 20125-39-7)

N6-(2-Phenylethyl)adenosine is a selective A1 adenosine receptor agonist with anti-proliferative activity on bladder cancer cells.

Chemical Structure

CAS 124555-18-6 GR 79236

Quick Inquiry

Verification code

Featured Items