GR 64349 - CAS 137593-52-3
Catalog number: B0084-165328
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C42H68N10O11S
Molecular Weight:
921.1147
COA:
Inquire
Targets:
Neurokinin Receptor
Description:
GR 64349 is a potent and selective agonist of tachykinin NK2 receptor (EC50 = 3.7 nM in rat colon).
Ordering Information
Catalog Number Size Price Stock Quantity
B0084-165328 1 mg $249 In stock
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Brife Description:
agonist of tachykinin NK2 receptor
Synonyms:
GR 64349; LYS-ASP-SER-PHE-VAL-GLY-R-GAMMA-LACTAM-LEU-MET-NH2; [LYS3, GLY8-R-GAMMA-LACTAM-LEU9]NEUROKININ A (3-10); L-Lys-L-Asp-L-Ser-L-Phe-L-Val-N-[(3R)-1-[(R)-1-[[[(S)-1-(Aminocarbonyl)-3-(methylthio)propyl]amino]carbonyl]-3-methylbutyl]-2-oxo-3α-pyrrolidi
Solubility:
Soluble to 1 mg/ml in water
MSDS:
Inquire
Density:
1.31g/cm3
InChIKey:
HVUNRXRFMQDMBO-NOJSRKIXSA-N
InChI:
InChI=1S/C42H68N10O11S/c1-23(2)19-32(40(61)46-27(35(45)56)15-18-64-5)52-17-14-28(42(52)63)47-41(62)34(24(3)4)51-38(59)29(20-25-11-7-6-8-12-25)49-39(60)31(22-53)50-37(58)30(21-33(54)55)48-36(57)26(44)13-9-10-16-43/h6-8,11-12,23-24,26-32,34,53H,9-10,13-22,43-44H2,1-5H3,(H2,45,56)(H,46,61)(H,47,62)(H,48,57)(H,49,60)(H,50,58)(H,51,59)(H,54,55)/t26-,27-,28-,29-,30-,31-,32-,34-/m0/s1
Canonical SMILES:
CC(C)CC(C(=O)NC(CCSC)C(=O)N)N1CCC(C1=O)NC(=O)C(C(C)C)NC(=O)C(CC2=CC=CC=C2)NC(=O)C(CO)NC(=O)C(CC(=O)O)NC(=O)C(CCCCN)N
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Chemical Structure

CAS 137593-52-3 GR 64349

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