GR 231118 - CAS 158859-98-4
Category: Inhibitor
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Neuropeptide Y receptor
GR 231118 is a potent neuropeptide Y (NPY) Y1 receptor antagonist (pA2 = 10 and 10.5 at rY1 and hY1 receptors, respectively) and an NPY Y4 receptor agonist (pEC50 = 6.0, 8.6 and 6.1 for rY2, hY4 and rY5 receptors, respectively). GR 231118 inhibits food intake in rats in vivo.
Brife Description:
NPY Y1 receptor antagonist, NPY Y4 receptor agonist
GR-231118; GR 231118; GR231118
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Chemical Structure

CAS 158859-98-4 GR 231118

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