GR 125487 sulfamate - CAS 859502-43-5
Category: Inhibitor
Please be kindly noted products are not for therapeutic use. We do not sell to patients.
Molecular Formula:
C19H26FN3O5S.H2NSO3H
Molecular Weight:
524.58
COA:
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Targets:
5-HT Receptor
Description:
GR 125487, a potent and selective 5-HT4 antagonist, is used in many biological assays to cross confirm the 5-HT4R agonist's activity.
Purity:
≥97% by HPLC
Related CAS:
859502-43-5 (Sulfmate); 144625-67-2 (Free Base)
Synonyms:
GR 125487 sulfamate; GR 125487; GR125487; GR-125487. 5-Fluoro-2-methoxy-[1-[2-[(methylsulfonyl)amino]ethyl]-4-piperidinyl]-1H-indole-3-methylcarboxylate sulfamate
Storage:
Store in a cool and dry place (or refer to the Certificate of Analysis).
MSDS:
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InChIKey:
LPMJZHPJOZETES-UHFFFAOYSA-M
InChI:
InChI=1S/C19H26FN3O5S.H3NO3S/c1-28-19-16(12-18(24)25)15-11-13(20)3-4-17(15)23(19)14-5-8-22(9-6-14)10-7-21-29(2,26)27;1-5(2,3)4/h3-4,11,14,21H,5-10,12H2,1-2H3,(H,24,25);(H3,1,2,3,4)/p-1
Canonical SMILES:
COC1=C(C2=C(N1)C=CC(=C2)F)C(=O)OCC3CCN(CC3)CCNS(=O)(=O)C.NS(=O)(=O)O
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CAS 859502-43-5 GR 125487 sulfamate

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