GNF-6231 - CAS 1243244-74-7
Catalog number: 1243244-74-7
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C25H28N6O2
Molecular Weight:
444.54
COA:
Inquire
Targets:
Others
Description:
This active molecular is a selective Porcupine protein inhibitor and IC50 value is 0.8nM. GNF-6231 shows efficient pathway inhibition and induced robust antitumor efficacy in animal tumor model. GNF-6231 may become a drug candidate for cancer treatment.
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Purity:
98%
Appearance:
Powder
Synonyms:
N-(5-(4-acetylpiperazin-1-yl)pyridin-2-yl)-2-(2',3-dimethyl-[2,4'-bipyridin]-5-yl)acetamide
Solubility:
Soluble in DMSO
Storage:
-20°C Freezer
MSDS:
Inquire
Application:
cancer treatment.
Quality Standard:
In-house standard
Shelf Life:
2 month in rt, long time
Quantity:
Milligrams-Grams
Canonical SMILES:
O=C(NC1=NC=C(N2CCN(C(C)=O)CC2)C=C1)CC3=CN=C(C4=CC(C)=NC=C4)C(C)=C3
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