Glutaminase C-IN-1 - CAS 311795-38-7
Catalog number:
311795-38-7
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C27H27BrN2O
Molecular Weight:
475.42
COA:
Inquire
Targets:
Others
Description:
Glutaminase C-IN-1, with effect to suppresse breast cancer cell growth and invasive activity in vitro, it is an allosteric, cell-permeable and reversible inhibitor of lutaminase C (IC50 = ~2.5 µM).
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Appearance:
Solid powder
Synonyms:
5-[3-bromo-4-(dimethylamino)phenyl]-2,2-dimethyl-1,3,5,6-tetrahydrobenzo[a]phenanthridin-4-one 5-(3-bromo-4-(dimethylamino)phenyl)-2,2-dimethyl-2,3,5,6-tetrahydrobenzo(a)phenanthridin-4(1H)-one
Solubility:
Soluble in DMSO
Storage:
Store in a cool and dry place and at 0 - 4℃ for short term (days to weeks) or -73℃ for long term (months to years).
MSDS:
Inquire
Shelf Life:
2 years
Boiling Point:
623.2±55.0 °C | Condition: Press: 760 Torr
Density:
1.39±0.1 g/cm3
InChIKey:
NVFRRJQWRZFDLM-UHFFFAOYSA-N
InChI:
1S/C27H27BrN2O/c1-27(2)14-19-24-18-8-6-5-7-16(18)9-11-21(24)29-26(25(19)23(31)15-27)17-10-12-22(30(3)4)20(28)13-17/h5-13,26,29H,14-15H2,1-4H3
Canonical SMILES:
CC1(CC2=C(C(NC3=C2C4=CC=CC=C4C=C3)C5=CC(=C(C=C5)N(C)C)Br)C(=O)C1)C
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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