|Description||Glisoxepide, a second-generation sulfonylurea, exerts greater binding affinity than the first-generation compounds. With antihyperglycemic activity, Glisoxepide is used as an antidiabetic drug used in the treatment of diabetes mellitus type 2.|
|Synonyms||N-[2-[4-[[[[(Hexahydro-1H-azepin-1-yl)amino]carbonyl]amino]sulfonyl]phenyl]ethyl]-5-methyl-3-isoxazolecarboxamide; 4-[4-[β-(5-Methylisoxazole-3-carboxamido)ethyl] phenylsulfonyl]-1,1-hexamethylenesemicarbazide; BS 4231; Glisepin; Glisoxepide; Pro-Diaban|
|Quantity||Data not available, please inquire.|
CP 81282 shows human renin and endothiapepsin inhibitory efficacy, but no detailed data has been published yet.
BIBF 1202 is the major in-vivo metabolite of BIBF 1120, which is an oral triple angiokinase inhibitor targeting VEGFR, PDGFR, FGFR. It is a related compound of ...
Erythromycin Ethylsuccinate, an oral macrolide antibiotic produced by Streptomyces erythreus, reversibly binds to the 50S ribosome of bacteria, and inhibits pro...
Omeprazole sulphone is the major metabolite of omeprazole, which is the gastric proton pump inhibitor. It is produced by cytochrome P450 (CYP)3A4 sulfoxidation ...
Amitraz is a non-systemic acaricide and insecticide, as an antiparasitic used to control red spider mites, leaf miners and scale insects.
Erdosteine is a mucolytic which is used in treatment of excessive viscous mucus.
XEN445 is a potent and selective endothelial lipase inhibitor with IC50 of 0.237 μM.
CVT10216 is a potent and selective, reversible inhibitor of aldehyde dehydrogenase 2 (ALDH2) with IC50 value of 29nM, thereby inhibiting dopamine synthesis. It ...
Schisanhenol, isolated from Schisandra rubriflora, has antioxidative effect on human LDL oxidation. The mechanism of Schisanhenol against LDL oxidation may be t...
Notoginsenoside R1 is extracted from the roots of Panax notoginseng (Burk.)F.H.Chen. It has some neuronal protective, antihypertensive effects and exhibits anti...
NSC134754 is a Heat Shock Factor 1 (HSF1) inhibitor. It can induce inhibition of HSF1, SP1 and NF-κB triggers the loss of the natural killer cell-activating lig...
Aucubin is an iridoid glycoside with a wide range of biological activities, including anti-inflammatory, anti-microbial, anti-algesic as well as anti-tumor acti...
Schisandrin B(Wuweizisu-B) is a dibenzocyclooctadiene derivative isolated from Fructus Schisandrae, has been shown to produce antioxidant effect on rodent liver...
Oct4 is a transcription factor which is involved in the reprogramming of somatic cells to produce pluripotent stem cells.
(-)-Epigallocatechin is the most abundant flavonoid in green tea. It is a major green tea polyphenol with antioxidant, anti-inflammatory, and anticancer activit...
Epothilone F, an active metabolite of Epothilone D, prevents cancer cells from dividing by interfering with tubulin.
Thiamet G is a potent, selective O-GlcNAcase inhibitor with Kiof 21 nM, while exhibiting 37,000-fold selectivity over human lysosomal –hexosaminidase.
Bisdemethoxycurcumin is one of the three major forms of curcuminoids found in the rhizomes of turmeric. Bisdemethoxycurcumin displays antioxidant, anti-inflamma...
LY 249933 is a bio-active molecular under the development of Eli Lilly. It has positive inotropic activity as a cardioselective 1,4-dihydropyridine compound.
Cetrimonium Bromide is a known component of the broad-spectrum antiseptic cetrimide, which is a mixture of different quaternary ammonium salts.