Givinostat hydrochloride - CAS 199657-29-9
Catalog number:
199657-29-9
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C24H28ClN3O4
Molecular Weight:
457.95
COA:
Inquire
Targets:
HDAC
Description:
Givinostat hydrochloride is the hydrochloride salt form of Givinostat. Givinostat, also called as GVS or ITF2357, a potent HDAC inhibitor for Maize HD2 (IC50= 10 nM), HD1-B (IC50= 7.5 nM nM) and HD1-A (IC50= 16 nM), has antiproliferative and proapoptotic
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Related CAS:
497833-27-9 (Free base); 732302-99-7 (HCl hydrate)
Appearance:
Solid powder
Synonyms:
(6-((diethylamino)methyl)naphthalen-2-yl)methyl (4-(hydroxycarbamoyl)phenyl)carbamate hydrochloride; ITF2357; ITF-2357; ITF 2357; ITF2357 HCl; ITF2357 hydrochloride; Givinostat HCl gavinostat,
Solubility:
Soluble in DMSO
Storage:
Store in a cool and dry place and at 0 - 4℃ for short term (days to weeks) or -33℃ for long term (months to years).
MSDS:
Inquire
Shelf Life:
2 years
InChIKey:
QKSGNWJOQMSBEP-UHFFFAOYSA-N
InChI:
1S/C24H27N3O4.ClH/c1-3-27(4-2)15-17-5-7-21-14-18(6-8-20(21)13-17)16-31-24(29)25-22-11-9-19(10-12-22)23(28)26-30;/h5-14,30H,3-4,15-16H2,1-2H3,(H,25,29)(H,26,28);1H
Canonical SMILES:
O=C(OCC1=CC=C2C=C(CN(CC)CC)C=CC2=C1)NC3=CC=C(C(NO)=O)C=C3.[H]Cl
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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