Gedatolisib (PF-05212384, PKI-587) - CAS 1197160-78-3
Catalog number: 1197160-78-3
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C32H41N9O4
Molecular Weight:
615.73
COA:
Inquire
Targets:
mTOR
Description:
Gedatolisib (PF-05212384, PKI-587) is a highly potent dual inhibitor of PI3Kα, PI3Kγ and mTOR with IC50 of 0.4 nM, 5.4 nM and 1.6 nM, respectively. Phase 2.
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Purity:
>98%
Synonyms:
N/A
MSDS:
Inquire
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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CAS 1197160-78-3 Gedatolisib (PF-05212384, PKI-587)

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