GDC-0084 - CAS 1382979-44-3
Catalog number:
1382979-44-3
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C18H22N8O2
Molecular Weight:
382.19
COA:
Inquire
Targets:
mTOR | PI3K
Description:
GDC-0084, a PI3K inhibitor, has been found to have probable antineoplastic effect and could pass blood-brain barrier with favourable penetration. It was just licensed to Novogen and start a Phase II trial for Glioma.
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Purity:
98%
Appearance:
Powder
Synonyms:
GDC-0084; 5-(6,6-dimethyl-4-morpholin-4-yl-8,9-dihydropurino[8,9-c][1,4]oxazin-2-yl)pyrimidin-2-amine
Solubility:
DMSO: ≥ 6 mg/mL
Storage:
-20ºC Freeze
MSDS:
Inquire
Application:
GDC-0084 is a PI3K inhibitor that has been found to have probable antineoplastic effect and could pass blood-brain barrier with favourable penetration.
Shelf Life:
As supplied, 2 years from the QC date provided on the Certificate of Analysis, when stored properly
Quantity:
Milligrams-Grams
InChIKey:
LGWACEZVCMBSKW-UHFFFAOYSA-N
InChI:
InChI=1S/C18H22N8O2/c1-18(2)16-22-12-14(25-3-6-27-7-4-25)23-13(11-9-20-17(19)21-10-11)24-15(12)26(16)5-8-28-18/h9-10H,3-8H2,1-2H3,(H2,19,20,21)
Canonical SMILES:
CC1(C2=NC3=C(N2CCO1)N=C(N=C3N4CCOCC4)C5=CN=C(N=C5)N)C
Current Developer:
Novogen
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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