Gaboxadol - CAS 64603-91-4
Catalog number:
64603-91-4
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C6H8N2O2
Molecular Weight:
140.14
COA:
Inquire
Targets:
GABA Receptor
Description:
Gaboxadol is a GABA agonist. It was a non-opioid analgesic and a novel type of hypnotic. It was first synthesized in 1977 by the Danish chemist Povl Krogsgaard-Larsen. It is an experimental sleep aid drug developed by Lundbeck and Merck. It was used as an analgesic and anxiolytic, as well as a treatment for tardive dyskinesia, Huntington's disease, Alzheimer's disease, and spasticity. It was in clinic phase 3 trials, but now it was terminated.
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Purity:
98%
Appearance:
White solid
Synonyms:
OV-101;Lu-02-030;MK-0928;Lu-02030;MK0928;Lu02030;THIP;4,5,6,7-Tetrahydroisoxazolo(5,4-c)pyridin-3(2H)-one;4,5,6,7-Tetrahydro-[1,2]oxazolo[5,4-c]pyridin-6-ium-3-one
Solubility:
Ethanol: 0.91 mg/mL
Storage:
-20°C Freezer
MSDS:
Inquire
Application:
Gaboxadol was used as an analgesic and anxiolytic, as well as a treatment for tardive dyskinesia, Huntington's disease, Alzheimer's disease, and spasticity.
Quality Standard:
In-house standard
Quantity:
Grams to Kilograms
Density:
1.36±0.1 g/cm3 | Condition: Temp: 20 °C Press: 760 Torr
InChIKey:
ZXRVKCBLGJOCEE-UHFFFAOYSA-O
InChI:
InChI=1S/C6H8N2O2/c9-6-4-1-2-7-3-5(4)10-8-6/h7H,1-3H2,(H,8,9)/p+1
Canonical SMILES:
C1C[NH2+]CC2=C1C(=O)NO2
Current Developer:
Gaboxadol was first synthesized in 1977 by the Danish chemist Povl Krogsgaard-Larsen. It is an experimental sleep aid drug developed by Lundbeck and Merck. It was in clinic phase 3 trials, but now it was terminated.
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CAS 64603-91-4 Gaboxadol

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