FRG8701 - CAS 108498-50-6
Category: Inhibitor
Please be kindly noted products are not for therapeutic use. We do not sell to patients.
Molecular Formula:
C22H30N2O4S
Molecular Weight:
418.55
COA:
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Targets:
Histamine Receptor
Description:
FRG-8701 is a novel Histamine H2 receptor antagonist (IC50= 0.25~ 0.43 μM). FRG-8701 has relatively long-lasting antisecretory ef fects in comparison with famotidine and cimetidine.
Synonyms:
FRG8701;FRG 8701; FRG-8701; 2-(furan-2-ylmethylsulfinyl)-N-[3-[3-(piperidin-1-ylmethyl)phenoxy]propyl]acetamide; FRG 8701; FRG-8701; N-(3-(3-(piperidinylmethyl)phenoxy)propyl)-2-(furfurylsulfinyl)acetamide
Storage:
Store in a cool and dry place (or refer to the Certificate of Analysis).
MSDS:
Inquire
Boiling Point:
675.2±55.0 ℃ at 760 Torr
Density:
1.226±0.06 g/cm3
InChIKey:
IWLUMUDDKHJJPB-UHFFFAOYSA-N
InChI:
1S/C22H30N2O4S/c25-22(18-29(26)17-21-9-5-13-28-21)23-10-6-14-27-20-8-4-7-19(15-20)16-24-11-2-1-3-12-24/h4-5,7-9,13,15H,1-3,6,10-12,14,16-18H2,(H,23,25)
Canonical SMILES:
C1CCN(CC1)CC2=CC(=CC=C2)OCCCNC(=O)CS(=O)CC3=CC=CO3
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Chemical Structure

CAS 108498-50-6 FRG8701

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