FR 113680 - CAS 126088-92-4
Catalog number: 126088-92-4
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C35H39N5O6
Molecular Weight:
625.72
COA:
Inquire
Targets:
Neurokinin 1 Receptor
Description:
FR 113680 is a novel tripeptide substance P antagonist with NK1 receptor selectivity originated by Fujisawa for the treatment of Asthma. But no development are reported yet.
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Purity:
98%
Appearance:
Powder
Synonyms:
Ac-Thr-trp(cho)-phe-N-mebzl;N-acetyl-L-threonyl-1-formyl-D-tryptophyl-N-methyl-N-(phenylmethyl)-L-Phenylalaninamide
Solubility:
Soluble in DMSO
Storage:
-20°C Freezer
MSDS:
Inquire
Application:
Asthma
Quality Standard:
In-house standard
Shelf Life:
2 month in rt, long time
Quantity:
Milligrams-Grams
InChIKey:
GUMFSDXELXANKA-KGLGFYCJSA-N
InChI:
1S/C35H39N5O6/c1-23(42)32(37-24(2)43)35(46)40(33(44)29(36)19-27-21-39(22-41)30-17-11-10-16-28(27)30)34(45)31(18-25-12-6-4-7-13-25)38(3)20-26-14-8-5-9-15-26/h4-17,21-23,29,31-32,42H,18-20,36H2,1-3H3,(H,37,43)/t23-,29-,31+,32+/m1/s1
Canonical SMILES:
C([C@@H]([N@@](Cc1ccccc1)C)Cc1ccccc1)(=O)N(C([C@H](N)Cc1cn(c2ccccc12)C=O)=O)C([C@@H](NC(=O)C)[C@@H](C)O)=O
Current Developer:
Originator: Fujisawa
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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