|Description||Fevipipran is a reversible competitive CRTh2 antagonist with IC50 value of 0.44 nM for inhibition of PGD2-induced eosinophil shape change in human whole blood. Now it is in Phase III clinical trials for the treatment of asthma.|
|Synonyms||NVP-QAW-039 QAW-039; 2-(2-methyl-1-(4-(methylsulfonyl)-2-(trifluoromethyl)benzyl)-1H-pyrrolo[2,3-b]pyridin-3-yl)acetic acid|
|Solubility||Soluble in DMSO|
|Application||Allergic asthma; Atopic dermatitis|
|Quality Standard||In-house standard|
|Shelf Life||2 month in rt, long tim|
|Current Developer||Originator Novartis|
This active molecular is a prostaglandin receptor agonist and detailed information has not been published yet.
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