Fasitibant chloride hydrochloride - CAS 869880-33-1
Catalog number:
869880-33-1
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C36-H49-Cl2-N6-O6-S.Cl-H.Cl
Molecular Weight:
836.71
COA:
Inquire
Targets:
Bradykinin Receptor
Description:
Fasitibant chloride is a selective nonpeptide kinin B2 receptor antagonist. Phase II clinical trials for the treatment of Osteoarthritis were discontinued.
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Purity:
98%
Appearance:
Powder
Synonyms:
MEN 16132; (S)-4-amino-5-(4-(4-((2,4-dichloro-3-(((2,4-dimethylquinolin-8-yl)oxy)methyl)phenyl)sulfonamido)tetrahydro-2H-pyran-4-carbonyl)piperazin-1-yl)-N,N,N-trimethyl-5-oxopentan-1-aminium chloride hydrochloride;1157852-02-2(Fasitibant chloride)
Solubility:
Soluble in DMSO
Storage:
-20℃ Freezer
MSDS:
Inquire
Application:
Osteoarthritis
Quality Standard:
In-house standard
Shelf Life:
2 month in rt, long time
Quantity:
Milligrams-Grams
InChIKey:
QIAWOUUTKDMGTE-UJXPALLWSA-M
InChI:
1S/C36H49Cl2N6O6S.2ClH/c1-24-22-25(2)40-33-26(24)8-6-10-30(33)50-23-27-28(37)11-12-31(32(27)38)51(47,48)41-36(13-20-49-21-14-36)35(46)43-17-15-42(16-18-43)34(45)29(39)9-7-19-44(3,4)5;;/h6,8,10-12,22,29,41H,7,9,13-21,23,39H2,1-5H3;2*1H/q+1;;/p-1/t29-;;/m0../s1
Canonical SMILES:
Cl.[Cl-].Cc1cc(C)c2cccc(OCc3c(Cl)ccc(c3Cl)S(=O)(=O)NC4(CCOCC4)C(=O)N5CCN(CC5)C(=O)[C@@H](N)CCC[N+](C)(C)C)c2n1
Current Developer:
Originator Menarini
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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