Fandosentan potassium - CAS 221246-12-4
Catalog number: 221246-12-4
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C25H17F3NO6S. K
Molecular Weight:
555.56
COA:
Inquire
Targets:
Endothelin Receptor
Description:
Fandosentan potassium is an endothelin A antagonist developed for the treatment of pulmonary hypertension.
Purity:
>98%
Appearance:
White to off-white crystalline powder
Synonyms:
potassium;4-(7-ethyl-1,3-benzodioxol-5-yl)-1,1-dioxo-2-[2-(trifluoromethyl)phenyl]-1$l^{6},2-benzothiazine-3-carboxylate; CI-1034; CI1034; PD 180988; PD180988
MSDS:
Inquire
Boiling Point:
387.9ºC at 760 mmHg
Melting Point:
235ºC
Density:
1.39 g/cm3
InChIKey:
MZWCHWWQSPPZRH-UHFFFAOYSA-M
InChI:
1S/C25H18F3NO6S.K/c1-2-14-11-15(12-19-23(14)35-13-34-19)21-16-7-3-6-10-20(16)36(32,33)29(22(21)24(30)31)18-9-5-4-8-17(18)25(26,27)28;/h3-12H,2,13H2,1H3,(H,30,31);/q;+1/p-1
Canonical SMILES:
CCC1=C2C(=CC(=C1)C3=C(N(S(=O)(=O)C4=CC=CC=C43)C5=CC=CC=C5C(F)(F)F)C(=O)[O-])OCO2.[K+]
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CAS 221246-12-4 Fandosentan potassium

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