Eribaxaban - CAS 536748-46-6
Catalog number:
536748-46-6
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C24H22ClFN4O4
Molecular Weight:
484.91
COA:
Inquire
Targets:
Factor Xa
Description:
Eribaxaban is an orally active inhibitor of coagulation factor Xa (activated factor X). It has anticoagulant activity and is used as an anticoagulant drug. It is used for the treatment and prevention of thrombotic disorders. It inhibited arterial thrombosis comparable to aspirin plus clopidogrel. It was developed by Pfizer. It was in phase II clinical trials, but has been terminated.
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Purity:
98%
Appearance:
Solid powder
Synonyms:
PD-0348292;PD0348292;(2R,4R)-N1-(4-Chlorophenyl)-N2-(2-fluoro-4-(2-oxopyridin-1(2H)-yl)phenyl)-4-methoxypyrrolidine-1,2-dicarboxamide
Solubility:
Soluble in DMSO, not in water
Storage:
-20°C Freezer
MSDS:
Inquire
Application:
Eribaxaban has anticoagulant activity and is used as an anticoagulant drug. It is used for the treatment and prevention of thrombotic disorders.
Quality Standard:
In-house standard
Quantity:
Milligrams-Grams
Density:
1.44±0.1 g/cm3 | Condition: Temp: 20 °C Press: 760 Torr
InChIKey:
QQBKAVAGLMGMHI-WIYYLYMNSA-N
InChI:
InChI=1S/C24H22ClFN4O4/c1-34-18-13-21(30(14-18)24(33)27-16-7-5-15(25)6-8-16)23(32)28-20-10-9-17(12-19(20)26)29-11-3-2-4-22(29)31/h2-12,18,21H,13-14H2,1H3,(H,27,33)(H,28,32)/t18-,21-/m1/s1
Canonical SMILES:
COC1CC(N(C1)C(=O)NC2=CC=C(C=C2)Cl)C(=O)NC3=C(C=C(C=C3)N4C=CC=CC4=O)F
Current Developer:
Eribaxaban was developed by Pfizer. It was in phase II clinical trials, but has been terminated.
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CAS 536748-46-6 Eribaxaban

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