|Description||EPZ015866，also called as GSK591, is a chemical probe for PRMT5 which has a role in diverse cellular processes including tumorigenesis. It exhibits excellent selectivity against a panel of methyltransferases. Inhibits the PRMT5/MEP50 complex from methylati|
|B0084-474632||300 mg||$499||In stock|
|Synonyms||2-(cyclobutylamino)-N-[(2S)-3-(3,4-dihydro-1H-isoquinolin-2-yl)-2-hydroxypropyl]pyridine-4-carboxamide EPZ015866 GSK591 GTPL8954 SCHEMBL16220740 GSK3203591 2-(cyclobutylamino)-N-[(2S)-2-hydroxy-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]pyridine-4-carbo|
|Solubility||DMSO,76 mg/mL (199.74 mM); Ethanol, 76 mg/mL (199.74 mM); Water, <1 mg/mL (<1 mM);|
|Storage||Store in a cool and dry place and at 0 - 4℃ for short term (days to weeks) or -28℃ for long term (months to years).|
|Shelf Life||2 years|
|Boiling Point||648.4±55.0 °C | Condition: Press: 760 Torr|
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