Enzalutamide - CAS 915087-33-1
Catalog number: B0084-155497
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C21H16F4N4O2S
Molecular Weight:
464.44
COA:
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Targets:
Androgen Receptor
Description:
Enzalutamide is an androgen-receptor (AR) antagonist with IC50 of 36 nM. It inhibits the activity of prostate cancer cell Ars, which over expressed in prostate cancer.
Ordering Information
Catalog Number Size Price Stock Quantity
B0084-155497 500 mg $199 In stock
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Brife Description:
androgen-receptor (AR) antagonist, prostate cancer
Purity:
>98%
Synonyms:
MDV3100; 4-(3-(4-cyano-3-(trifluoromethyl)phenyl)-5,5-dimethyl-4-oxo-2-thioxoimidazolidin-1-yl)-2-fluoro-N-methylbenzamide
MSDS:
Inquire
Application:
potential antineoplastic agent
InChIKey:
WXCXUHSOUPDCQV-UHFFFAOYSA-N
InChI:
InChI=1S/C21H16F4N4O2S/c1-20(2)18(31)28(12-5-4-11(10-26)15(8-12)21(23,24)25)19(32)29(20)13-6-7-14(16(22)9-13)17(30)27-3/h4-9H,1-3H3,(H,27,30)
Canonical SMILES:
CC1(C(=O)N(C(=S)N1C2=CC(=C(C=C2)C(=O)NC)F)C3=CC(=C(C=C3)C#N)C(F)(F)F)C
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CAS 915087-33-1 Enzalutamide

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