Enrasentan - CAS 167256-08-8
Catalog number: 167256-08-8
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C29H30O8
Molecular Weight:
506.55
COA:
Inquire
Targets:
Endothelin Receptor
Description:
Enrasentan, an indene derivative, has been found to be an endothelin receptor antagonist that was once studied in reperfusion injury and heart failure therapy.
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Purity:
98%
Appearance:
Powder
Synonyms:
Enrasentan; SB-217242; UNII-QG16H8A6ZH; SB 217242; CHEMBL431651; (1S,2R,3S)-1-(1,3-benzodioxol-5-yl)-3-[2-(2-hydroxyethoxy)-4-methoxyphenyl]-5-propoxy-2,3-dihydro-1H-indene-2-carboxylic acid
Storage:
Store in a cool and dry place and at 0 - 4 °C for short term (days to weeks) or -20 °C for long term (months to years).
MSDS:
Inquire
Quality Standard:
In-house standard
Quantity:
Milligram-Grams
InChIKey:
GLCKXJLCYIJMRB-UPRLRBBYSA-N
InChI:
InChI=1S/C29H30O8/c1-3-11-34-19-6-7-20-22(14-19)27(21-8-5-18(33-2)15-24(21)35-12-10-30)28(29(31)32)26(20)17-4-9-23-25(13-17)37-16-36-23/h4-9,13-15,26-28,30H,3,10-12,16H2,1-2H3,(H,31,32)/t26-,27+,28+/m0/s1
Canonical SMILES:
CCCOC1=CC2=C(C=C1)C(C(C2C3=C(C=C(C=C3)OC)OCCO)C(=O)O)C4=CC5=C(C=C4)OCO5
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