|Description||Endoxifen hydrochloride is a metabolite of Tamoxifen and a selective estrogen receptor modulator (SERM) that inhibits the growth of estrogen-stimulated BT474 cells (IC50 = 54 nM). Endoxifen is used for the treatment of estrogen receptor (ER) positive breast cancer.|
|Brife Description||SERM, breast cancer|
|Related CAS||112093-28-4 (free base)|
|Synonyms||4-[1-[4-[2-(methylamino)ethoxy]phenyl]-2-phenyl-1-buten-1-yl]-Phenol hydrochloride (1:1)|
Nafoxidine, a triphenylethylene nonsteroidal agent, is a partial estrogen antagonist.
Endoxifen E-isomer hydrochloride
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