Endoxifen - CAS 112093-28-4
Catalog number:
112093-28-4
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C25H27NO2
Molecular Weight:
373.49
COA:
Inquire
Targets:
Estrogen Receptor/ERR
Description:
Endoxifen, a significant metamolite of Tamoxifen, is a regulator of estrogen receptor and could be effective in the treatment of estrogen-dependent breast cancer. IC50: 1.6 μM.
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Purity:
>98 %
Appearance:
Off-White to Pink Solid
Synonyms:
4-[(1Z)-1-[4-[2-(Methylamino)ethoxy]phenyl]-2-phenyl-1-buten-1-yl]phenol;
Solubility:
10 mM in DMSO
Storage:
Amber Vial, -86°C Freezer, Under Inert Atmosphere
MSDS:
Inquire
Application:
Endoxifen is a regulator of estrogen receptor and could be effective in the treatment of estrogen-dependent breast cancer.
Shelf Life:
As supplied, 2 years from the QC date provided on the Certificate of Analysis, when stored properly
Quantity:
Milligrams-Grams
Boiling Point:
519.327ºC at 760 mmHg
Density:
1.099g/cm3
InChIKey:
MHJBZVSGOZTKRH-IZHYLOQSSA-N
InChI:
InChI=1S/C25H27NO2/c1-3-24(19-7-5-4-6-8-19)25(20-9-13-22(27)14-10-20)21-11-15-23(16-12-21)28-18-17-26-2/h4-16,26-27H,3,17-18H2,1-2H3/b25-24-
Canonical SMILES:
CCC(=C(C1=CC=C(C=C1)O)C2=CC=C(C=C2)OCCNC)C3=CC=CC=C3
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CAS 112093-28-4 Endoxifen

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