Encaleret - CAS 787583-71-5
Catalog number: 787583-71-5
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C29H33ClFNO4
Molecular Weight:
514.03
COA:
Inquire
Targets:
CaSR
Description:
Encaleret is a calcium-sensing receptor (CaSR) antagonist. But in Oct 2011, Phase-II for Osteoporosis in USA was discontinued.
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Purity:
98%
Appearance:
Powder
Synonyms:
1214922-52-7 (sulfate salt);JIT-305;2'-((R)-1-((R)-3-((1-(4-chloro-3-fluorophenyl)-2-methylpropan-2-yl)amino)-2-hydroxypropoxy)ethyl)-3-methyl-[1,1'-biphenyl]-4-carboxylic acid
Solubility:
Soluble in DMSO
Storage:
-20℃ Freezer
MSDS:
Inquire
Application:
Osteoporosis
Quality Standard:
In-house standard
Shelf Life:
2 month in rt, long time
Quantity:
Milligrams-Grams
InChIKey:
UNFHDRVFEQPUEL-DENIHFKCSA-N
InChI:
InChI=1S/C29H33ClFNO4/c1-18-13-21(10-11-23(18)28(34)35)25-8-6-5-7-24(25)19(2)36-17-22(33)16-32-29(3,4)15-20-9-12-26(30)27(31)14-20/h5-14,19,22,32-33H,15-17H2,1-4H3,(H,34,35)/t19-,22-/m1/s1
Canonical SMILES:
CC1=C(C=CC(=C1)C2=CC=CC=C2C(C)OCC(CNC(C)(C)CC3=CC(=C(C=C3)Cl)F)O)C(=O)O
Current Developer:
Merck & Co
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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CAS 787583-71-5 Encaleret

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